Publications
6E11, a highly selective inhibitor of Receptor-Interacting Protein Kinase 1, protects cells against cold hypoxia-reoxygenation injury
Delehouze, C.; Leverrier-Penna, S.; Le Cann, F.; Comte, A.; Jacquard-Fevai, M.; Delalande, O.; Desban, N.; Baratte, B.; Gallais, I.; Faurez, F.; Bonnet, M.; Hauteville, M.; Goekjian, P.; Thuillier, R.; Favreau, F.; Vandenabeele, P.; Bach S.; Dimanche-Boitrel M. T.
Scientific Reports volume 7, Article number: 12931 (2017)
Sibiriline, a new small chemical inhibitor of receptor-interacting protein kinase 1, prevents immune-dependent hepatitis
Le Cann, F.; Delehouze, C.; Leverrier-Penna, S.; Filliol, A.; Comte, A.; Delalande, O.; Desban, N.; Baratte, B.; Gallais, I.; Piquet-Pellorce, C.; Faurez, F.; Bonnet, M.; Mettey, Y.; Goekjian, P.; Samson, M.; Vandenabeele, P.; Bach S.; Dimanche-Boitrel M. T.
FEBS J. 2017, 18, 3050-3068
Synthesis of 1-Indanols and 1-Indanamines by Intramolecular Palladium(0)-Catalyzed C(sp3)H Arylation: Impact of Conformational Effects
Janody, S.; Jazzar, R.; Comte, A.; Holstein, P. M.; Vors, J-P.; Ford, M. J.; Baudoin, O.
Chem. Eur. J. 2014, 20, 11084-11090
Synthesis of cyclobutarenes by palladium-catalyzed C(sp3)-H bond arylation: Preparation of methyl 7-methylbicyclo[4.2.0]octa-1,3,5-triene-7-carboxylate
Davi, M.; Comte, A.; Jazzar, R.; Baudoin, O.
Org. Synth. 2012, 89, 510-522
N,N’-alkylated Imidazolium-Derivatives Act as Quorum-Sensing Inhibitors Targeting the Pectobacterium atrosepticum-Induced Symptoms on Potato Tubers
Raoul des Essarts, Y.; Sabbah, M.; Comte, A.; Soulère, L.; Queneau, Y.; Hélias, V.; Faure, F.
Int. J. Mol. Sci. 2013, 14, 19976-19986
Structure–Activity Relationship of S-Trityl-l-Cysteine Analogues as Inhibitors of the Human Mitotic Kinesin Eg5
DeBonis, S.; Skoufias, D.A.; Indorato, R.-L.; Liger, F.; Marquet, B.; Laggner, C.; Joseph, B.; Kozielski, F.
J. Med. Chem. 2008, 51, 1115-1125
Meriolins (3-(Pyrimidin-4-yl)-7-azaindoles): Synthesis, Kinase Inhibitory Activity, Cellular Effects, and Structure of a CDK2/CyclinA/Meriolin Complex
Echalier, A.; Bettayeb, K.; Ferandin, Y.; Lozach, O.; Clement, M.; Valette, A.; Liger, F.;Marquet, B.; Morris, J.C.; Endicott, J.A.; Joseph, B.; Meijer, L.
J. Med. Chem. 2008, 51, 737-751
Meriolins, a New Class of CellDeath-Inducing Kinase Inhibitors with Enhanced Selectivity for Cyclin-Dependent Kinases
Bettayeb, K.; Tirado, O.M.; Marionneau-Lambot, S.; Ferandin, Y.; Lozach, O.; Morris, J.C.;Mateo-Lozano, S.; Drueckes, P.; Schaechtele, C.; Kubbutat, M.H.G.; Liger, F.; Marquet, B.;Joseph, B.; Echalier, A.; Endicott, J.A.; Notario, V.; Meijer, L.
Cancer Res. 2007, 67, 8325-8334
Synthesis and evaluation of new arylbenzo[b]thiophene and diarylthiophene derivatives as inhibitors of the NorA multidrug transporter of Staphylococcus aureus
Fournier Dit Chabert, J.; Marquez, B.; Neville, L.; Joucla, L.; Broussous, S.; Bouhours, P.; David, E.; Pellet-Rostaing, S.; Marquet, B.; Moreau, N.; Lemaire, M.